HCID 13608622, compound → HCID 131722952, compound

Participants

Reaction Steps

N-(4-Benzyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-ylylmethyl)-3-(1H-indol-3-yl)-butyramide. (4-Benzyl-3,4-dihydro-2H-benzo[1,4]oxazin-2-yl)-methylamnine (1.2 g, 4.7 mmol) was coupled to indole butyric acid (1.8 g, 8.9 mmol) according to the procedure used to prepare intermediatel 1 above to afford 1.3 g (63%) of the title compound as a yellow solid: mp 61-63.5° C.; MS (EI) m/e 439 (M+)

Provenance & Evidence