HRID446320

反应详情

EQUATION

反应方程式

HRID 446320 反应方程式

AUXILIARIES

试剂、催化剂与溶剂

1

CONDITIONS

反应条件

温度
80 °C

PROCEDURE

实验过程

To phenyl 3-methyl-4-(3-(2-(methylamino)pyrimidin-4-yl)pyridin-2-yloxy)phenylcarbamate (59 mg, 0.14 mmol) in THF (1 mL) was added 2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)benzenamine (30 mg, 0.12 mmol). The mixture was stirred for 40 hours at 80° C. The crude material was purified by silica gel chromatography (0-20% MeOH/CH2Cl2) to yield the title compound as a light yellow solid. MS m/z=593 [M+H]+. Calc'd for C30H31F3N8O2: 592.63.

WORKUP

后处理

  1. customThe crude material was purified by silica gel chromatography (0-20% MeOH/CH2Cl2)