Piperidin-4-ol → HCID 68577305, compound

HRID 446874Notes

Reaction equation

HRID 446874 reaction equation
[F:1][C:2]1[CH:31]=[CH:30][C:5]([O:6][C:7]2[CH:12]=[CH:11][CH:10]=[CH:9][C:8]=2[NH:13][S:14]([C:17]2[CH:29]=[CH:28][C:20]([C:21]([NH:23][CH2:24][C:25](O)=[O:26])=[O:22])=[CH:19][CH:18]=2)(=[O:16])=[O:15])=[CH:4][CH:3]=1.[OH:32][CH:33]1[CH2:38][CH2:37][NH:36][CH2:35][CH2:34]1>>[F:1][C:2]1[CH:31]=[CH:30][C:5]([O:6][C:7]2[CH:12]=[CH:11][CH:10]=[CH:9][C:8]=2[NH:13][S:14]([C:17]2[CH:18]=[CH:19][C:20]([C:21]([NH:23][CH2:24][C:25]([N:36]3[CH2:37][CH2:38][CH:33]([OH:32])[CH2:34][CH2:35]3)=[O:26])=[O:22])=[CH:28][CH:29]=2)(=[O:15])=[O:16])=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 79341Piperidin-4-olHCID 68577142HCID 68577142, compound

Product 1

HCID 68577305HCID 68577305, compound

Procedure

The title compound was prepared from {4-[2-(4-fluoro-phenoxy)-phenylsulfamoyl]-benzoylamino}-acetic acid and 4-hydroxypiperidine according to the method described in Example 1.1/f. MS (EI) 528.4 (MH+).

Sources & evidence

ORD record
ord-68b4aaa662ae416091671180cd504ba0
Source dataset
uspto-grants-2013_07
Patent number
US08481527B2

Reaction notes

Loading…