(4-Methoxyphenyl)boronic acid → HCID 86595320, compound

HRID 447200Notes

Reaction equation

HRID 447200 reaction equation
[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[NH:13][CH:14]=2)[CH:5]=[CH:4][N:3]=1.[CH3:16][O:17][C:18]1[CH:23]=[CH:22][C:21](B(O)O)=[CH:20][CH:19]=1>>[Cl:1][C:2]1[CH:7]=[C:6]([C:8]#[C:9][C:10]2[N:11]=[C:12]([CH3:15])[N:13]([C:21]3[CH:22]=[CH:23][C:18]([O:17][CH3:16])=[CH:19][CH:20]=3)[CH:14]=2)[CH:5]=[CH:4][N:3]=1

Participants

3

Reactant 2

HCID 201262(4-Methoxyphenyl)boronic acidHCID 178418879HCID 178418879, compound

Product 1

HCID 86595320HCID 86595320, compound

Procedure

The title compound, MS: m/e=324.8 (M+H+), was prepared in accordance with the general method of example 7 from 2-chloro-4-(2-methyl-1H-imidazol-4-ylethynyl)-pyridine and 4-methoxy-benzene boronic acid.

Sources & evidence

ORD record
ord-e3cced6c980749bc9bd7070d6ebdb661
Source dataset
uspto-grants-2013_07
Patent number
US08481548B2

Reaction notes

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