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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 449333Generated: October 29, 2026

4-(Methylcarbamoyl)benzeneboronic acid → 4-(6-fluoropyridin-3-yl)-N-methylbenzamide

https://huagongshe.com/reaction/449333

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(Methylcarbamoyl)benzeneboronic acidHCID 2773526—
Reactant5-Bromo-2-fluoropyridineHCID 2783168—
Product4-(6-fluoropyridin-3-yl)-N-methylbenzamideHCID 59496610—

Reaction Steps

This compound was prepared from 5-bromo-2-fluoropyridine and {4-[(methylamino)carbonyl]phenyl}boronic acid using procedures analogous to those for Example 18, step 1. Analytic LCMS (M+H)+: m/z=231.1.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08481732B2
Source datasetuspto-grants-2013_07
ORD IDord-34f54c66e3a9478eab1f60f71a582125
Source noteuspto-grants-2013_07