1-((2,4-Dichlorophenyl)methyl)-1H-pyrazol-3-amine → [1-(2,4-Dichloro-benzyl)-1H-pyrazol-3-yl]-[1-(3-methyl-[1,2,4]thiadiazol-5-yl)-piperidin-4-yl]-amine

Participants

Role	Name	HCID	Charge
Reactant	1-((2,4-Dichlorophenyl)methyl)-1H-pyrazol-3-amine	HCID 5302743	—
Reactant	1-(3-Methyl-1,2,4-thiadiazol-5-yl)piperidin-4-one	HCID 59258510	—
Product	[1-(2,4-Dichloro-benzyl)-1H-pyrazol-3-yl]-[1-(3-methyl-[1,2,4]thiadiazol-5-yl)-piperidin-4-yl]-amine	HCID 53354736	—

Reaction Steps

Prepared in analogy to example 1 step h) starting from 1-(3-methyl-[1,2,4]thiadiazol-5-yl)-piperidin-4-one (example 1c) and 1-(2,4-dichloro-benzyl)-1H-pyrazol-3-ylamine. The title compound was obtained as a colorless oil (yield=56%).

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US08486967B2
Source dataset	uspto-grants-2013_07
ORD ID	ord-0e95c66d07824572a5969d70c2e3b0c6
Source note	uspto-grants-2013_07