反应详情

Prepared in analogy to example 1 step h) starting from 1-(2-chloropyridin-4-yl)piperidin-4-one (see example 232b) and 8-(3-tert-butylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine. The latter compound can be prepared in analogy to example 1 steps d-f) starting from 2-amino-6-bromo-pyridine and 3-tert-butylphenylboronic acid (EP2243785A1). The title compound was obtained as a colourless foam. MS ISP (m/e): 461.2 [(M+H)+].

1. customPrepared in analogy to example 1 step h)
2. customThe latter compound can be prepared in analogy to example 1 steps d-f)