HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-Amino-6-bromopyridine → HCID 86656718, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-Amino-6-bromopyridine | HCID 300809 | — |
| Reactant | (3-tert-Butylphenyl)boronic acid | HCID 21582509 | — |
| Reactant | 8-(3-Tert-butylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine | HCID 67344991 | — |
| Reactant | 1-(2-Chloropyridin-4-yl)piperidin-4-one | HCID 86656719 | — |
| Product | HCID 86656718 | HCID 86656718 | — |
Reaction Steps
Prepared in analogy to example 1 step h) starting from 1-(2-chloropyridin-4-yl)piperidin-4-one (see example 232b) and 8-(3-tert-butylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine. The latter compound can be prepared in analogy to example 1 steps d-f) starting from 2-amino-6-bromo-pyridine and 3-tert-butylphenylboronic acid (EP2243785A1). The title compound was obtained as a colourless foam. MS ISP (m/e): 461.2 [(M+H)+].
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08486967B2 |
| Source dataset | uspto-grants-2013_07 |
| ORD ID | ord-e7ea2fad305b4862907c2491420b252e |
| Source note | uspto-grants-2013_07 |