1,4-Dioxane hydrochloride → 5-Benzoyloxy-2-aminoindan hydrochloride

Participants

Reaction Steps

Using 5-benzoyloxy-2-(tert-butoxycarbonylamino)indan (130 mg, 0.37 mmol), 4N hydrochloric acid-dioxane (2 ml) and acetic acid (6 ml), a similar procedure to Production Example 213 was carried out to obtain 5-benzoyloxy-2-aminoindan hydrochloride (67 mg, 0.35 mmol) having the following physical properties:

Provenance & Evidence