HuagongsheHuagongshe Chemistry Print Report · For research reference only
HCID 57963062, compound → HCID 67200711, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | HCID 57963062 | HCID 57963062 | — |
| Reactant | 1H-Pyrrolo[2,3-b]pyridine, 3-iodo-5-methoxy-1-(phenylsulfonyl)- | HCID 59128707 | — |
| Product | HCID 67200711 | HCID 67200711 | — |
Reaction Steps
(5-Fluoro-2-methoxy-pyridin-3-ylmethyl)-[5-(5-methoxy-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-pyrimidin-2-yl]-amine P-1599 is prepared in three steps from 1-benzenesulfonyl-3-iodo-5-methoxy-1H-pyrrolo[2,3-b]pyridine 16 and (5-fluoro-2-methoxy-pyridin-3-ylmethyl)-(5-formyl-pyrimidin-2-yl)-carbamic acid tert-butyl ester 123 as shown in Scheme 13.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09096593B2 |
| Source dataset | uspto-grants-2015_08 |
| ORD ID | ord-f9be122e05434f3381e54f545d409aae |
| Source note | uspto-grants-2015_08 |