反应详情

In a similar fashion using route 14 general procedure 26, 5-chloroquinolin-8-amine (Intermediate 27) (50 mg, 0.28 mmol), 2,4-dichlorobenzenesulfonyl chloride (103 mg, 0.42 mmol) gave the title compound (40 mg, 40%) after purification by column chromatography with DCM as the eluent.