HCID 68639572, compound → HCID 86732324, compound

Participants

Reaction Steps

The title compound is prepared in analogy to 4-(4-bromo-2-(methylsulfonyl)phenyl)-1-(3-(trifluoromethyl)phenyl)-3,4,7,8-tetrahydroquinazoline-2,5(1H,6H)-dione (intermediate 34), using 1-(3-(difluoromethyl)phenyl)urea (intermediate 35, 707 mg, 3.80 mmol) as starting material. Yield: 319 mg; ESI mass spectrum [(79Br)-M+H]+=525, [(81Br)-M+H]+=527, Retention time HPLC: 1.01 min (Z017_S04).

Provenance & Evidence