HuagongsheHuagongshe Chemistry Print Report · For research reference only
Acetic Acid → N2 (Diphenylacetyl)-N-[(1H-indol-5-yl) methyl]-argininamide acetate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Acetic Acid | HCID 176 | — |
| Reactant | HCID 136381104 | HCID 136381104 | — |
| Catalyst | Palladium | HCID 23938 | — |
| Product | N2 (Diphenylacetyl)-N-[(1H-indol-5-yl) methyl]-argininamide acetate | HCID 178476730 | 54% |
Reaction Steps
Prepared analogously to Example 1c) from N5 -[amino(nitroimino)methyl]-N2 -(diphenylacetyl)-N-[(1H-indol-5-yl)methyl]-ornithinamide by catalytic hydrogenation in the presence of palladium black and 80% aqueous acetic acid in a yield of 54% of theory.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US05616620 |
| Source dataset | uspto-grants-1997_04 |
| ORD ID | ord-bc7c2b265dab44cf8d65451939da42e6 |
| Source note | uspto-grants-1997_04 |