6-Methoxy-3-pyridinylamine → HCID 178471949, compound

HRID 526259Notes

Reaction equation

HRID 526259 reaction equation
[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:6]([NH2:9])=[CH:5][N:4]=1.C(O[CH:13]=[C:14]([C:20](=[O:24])[CH:21]([CH3:23])[CH3:22])[C:15]([O:17][CH2:18][CH3:19])=[O:16])C>>[CH3:1][O:2][C:3]1[N:4]=[CH:5][C:6]([NH:9][CH:13]=[C:14]([C:20](=[O:24])[CH:21]([CH3:23])[CH3:22])[C:15]([O:17][CH2:18][CH3:19])=[O:16])=[CH:7][CH:8]=1

Participants

3

Reactant 2

HCID 811216-Methoxy-3-pyridinylamineHCID 54219628HCID 54219628, compound

Product 1

HCID 178471949HCID 178471949, compound

Procedure

Ethyl 2-(((6-methoxypyridin-3-yl)amino)methylene)-4-methyl-3-oxopentanoate was prepared with conditions described in Example 99 using 2-methoxy-5-aminopyridine and ethyl 2-(ethoxymethylene)-4-methyl-3-oxopentanoate.

Sources & evidence

ORD record
ord-63b637e15b69487e8aa80f881e96d0dc
Source dataset
uspto-grants-2016_05
Patent number
US09345709B2

Reaction notes

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