HCID 118524119, compound → HCID 118524034, compound

Participants

Reaction Steps

Using similar reaction conditions as described in step-ii of example-7, tert-butyl 4-(4-(3-(1-(3-fluorobenzyl)-1H-pyrazol-4-yl)-1-tosyl-1H-pyrrolo[2,3-b]pyridin-5-yl)phenyl)-1,4-diazepane-1-carboxylate (120 mg, 0.166 mmol) was deprotected in TFA/DCM (3/1 ml) to afford 100 mg (97.0% yield) of the titled compound. MS: m/z=621.2 (M+1).

Provenance & Evidence