2-Morpholinoethylamine → HCID 66998257, compound

HRID 559225Notes

Reaction equation

[Cl:1][CH2:2][C:3]1[N:7]([CH3:8])[N:6]=[C:5]([C:9]2[CH:10]=[C:11]3[C:15](=[CH:16][CH:17]=2)[N:14]([CH3:18])[C:13]2[N:19]([CH3:32])[C:20](=[O:31])[C:21]([C:23]4[CH:28]=[CH:27][C:26]([Cl:29])=[CH:25][C:24]=4[Cl:30])=[CH:22][C:12]3=2)[CH:4]=1.[NH2:33][CH2:34][CH2:35][N:36]1[CH2:41][CH2:40][O:39][CH2:38][CH2:37]1>>[ClH:1].[Cl:30][C:24]1[CH:25]=[C:26]([Cl:29])[CH:27]=[CH:28][C:23]=1[C:21]1[C:20](=[O:31])[N:19]([CH3:32])[C:13]2[N:14]([CH3:18])[C:15]3[C:11]([C:12]=2[CH:22]=1)=[CH:10][C:9]([C:5]1[CH:4]=[C:3]([CH2:2][NH:33][CH2:34][CH2:35][N:36]2[CH2:41][CH2:40][O:39][CH2:38][CH2:37]2)[N:7]([CH3:8])[N:6]=1)=[CH:17][CH:16]=3

Participants

Reactant 2

HCID 4082852-Morpholinoethylamine

HCID 66997926HCID 66997926, compound

Product 1

HCID 66998257HCID 66998257, compound

Procedure

The process is carried out as in Example 122 above, with the compound from Example 122A: 6-(5-chloromethyl-1-methyl-1H-pyrazol-3-yl)-3-(2,4-dichloro-phenyl)-1,9-dimethyl-1,9-dihydropyrido[2,3-b]indol-2-one and aminoethyl-morpholine.

Sources & evidence

ORD record: ord-7c58e3d298574d5084e1b7c972a489f5
Source dataset: uspto-grants-2011_11
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US08063061B2

Reaction notes

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