Cyclobutanone → HCID 59197916, compound

HRID 560214Notes

Reaction equation

[N:1]1([C:6]2([C:10]#[N:11])[CH2:9]O[CH2:7]2)[CH2:5][CH2:4][CH2:3][CH2:2]1.[C:12]1(=O)CCC1.[CH:17]1([N:20]2CCNCC2)[CH2:19][CH2:18]1>>[CH:17]1([N:20]2[CH2:4][CH2:5][N:1]([C:6]3([C:10]#[N:11])[CH2:9][CH2:12][CH2:7]3)[CH2:2][CH2:3]2)[CH2:19][CH2:18]1

Participants

Reactant 3

HCID 14496Cyclobutanone

HCID 47420041-Cyclopropylpiperazine

HCID 591979193-Cyano-3-(pyrrolidin-1-YL)oxetane

Product 1

HCID 59197916HCID 59197916, compound

Procedure

The title compound, colourless oil, MS: m/e=179.1 [(M−CN)+], was prepared in accordance with the general method of intermediate A from cyclobutanone and 1-cyclopropyl-piperazine.

Sources & evidence

ORD record: ord-84c1d57757f24dcf8228d0a931c2f9a0
Source dataset: uspto-grants-2011_11
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US08063098B2

Reaction notes

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