HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acid → 2-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-5'-ethoxycarbonylmethyl-2'-methoxy-biphenyl-4-carboxylic acid
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acid | HCID 57419864 | — |
| Reactant | [4-Methoxy-3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-acetic acid ethyl ester | HCID 58120060 | — |
| Product | 2-[(Benzyloxycarbonyl-ethyl-amino)-methyl]-5'-ethoxycarbonylmethyl-2'-methoxy-biphenyl-4-carboxylic acid | HCID 54674329 | — |
Reaction Steps
Prepared according to the procedure described in Example 1, Step 4, using the following starting materials: 3-[(benzyloxycarbonyl-ethyl-amino)-methyl]-4-bromo-benzoic acid and [4-methoxy-3-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-acetic acid ethyl ester. M+H is 506.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08067445B2 |
| Source dataset | uspto-grants-2011_11 |
| ORD ID | ord-eee2d4fd3ba3495cbf08131f2075c95f |
| Source note | uspto-grants-2011_11 |