Methylamine → HCID 178482442, compound

Participants

Reaction Steps

2-Dimethylamino-5-[1-(6-fluoroindol-3-yl)ethyl]-2-oxazolin-4-one (340 mg) was dissolved into methylamine (5 ml) at −10° C. The mixture was stirred for 3 hours at the same temperature. The mixture was concentrated to give a residue, which was subjected to column chromatography. Elution with hexane-acetone (1:1) provided the titled compound (254 mg).

Provenance & Evidence