3,3-Diphenylpropylamine → HCID 131722264, compound

HRID 565658Notes

Reaction equation

HRID 565658 reaction equation
[CH:1]([CH2:3][CH:4]1[CH2:9][CH2:8][N:7]([CH2:10][C:11]2([CH3:31])[CH2:15][C:14]3[C:16]([CH3:30])=[C:17]([NH:22][C:23](=[O:29])[O:24][C:25]([CH3:28])([CH3:27])[CH3:26])[C:18]([CH3:21])=[C:19]([CH3:20])[C:13]=3[O:12]2)[CH2:6][CH2:5]1)=O.[C:32]1([CH:38]([C:42]2[CH:47]=[CH:46][CH:45]=[CH:44][CH:43]=2)[CH2:39][CH2:40][NH2:41])[CH:37]=[CH:36][CH:35]=[CH:34][CH:33]=1>>[C:42]1([CH:38]([C:32]2[CH:33]=[CH:34][CH:35]=[CH:36][CH:37]=2)[CH2:39][CH2:40][NH:41][CH2:1][CH2:3][CH:4]2[CH2:9][CH2:8][N:7]([CH2:10][C:11]3([CH3:31])[CH2:15][C:14]4[C:16]([CH3:30])=[C:17]([NH:22][C:23](=[O:29])[O:24][C:25]([CH3:28])([CH3:27])[CH3:26])[C:18]([CH3:21])=[C:19]([CH3:20])[C:13]=4[O:12]3)[CH2:6][CH2:5]2)[CH:43]=[CH:44][CH:45]=[CH:46][CH:47]=1

Participants

3

Reactant 2

HCID 796983,3-DiphenylpropylamineHCID 53952919HCID 53952919, compound

Product 1

HCID 131722264HCID 131722264, compoundYield 97%

Procedure

Using tert-butyl [2-[[4-(formylmethyl)-1-piperidinyl]methyl]-2,3-dihydro-2,4,6,7-tetramethylbenzofuran-5yl]carbamate and (3,3-diphenylpropyl)amine, the procedure of Reference Example 44 was otherwise repeated to provide the title compound. Yield 97%.

Sources & evidence

ORD record
ord-4db9a36ad1d948c28eecd319978805b3
Source dataset
uspto-grants-2001_01
Patent number
US06172085B2

Reaction notes

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