6,7-Dihydro-5H-pyrrolo[3,4-b]pyridine hydrochloride → 3-[(4-(5H-Pyrrolo[3,4-b]pyridin-6(7H)-yl)-1,3,5-triazin-2-yl)amino]-benzenemethanesulfonamide

Participants

Role	Name	HCID	Charge
Reactant	6,7-Dihydro-5H-pyrrolo[3,4-b]pyridine hydrochloride	HCID 18953643	—
Reactant	3-[(4-Chloro-1,3,5-triazin-2-yl)amino]benzenemethanesulfonamide	HCID 86679822	—
Product	3-[(4-(5H-Pyrrolo[3,4-b]pyridin-6(7H)-yl)-1,3,5-triazin-2-yl)amino]-benzenemethanesulfonamide	HCID 60197808	—

Reaction Steps

B48 was prepared following the general procedure reported for B10 using A1 and 6,7-dihydro-5H-pyrrolo[3,4-b]pyridine hydrochloride; yield: 92.2 mg (24%), dark amorphous solid. MS (ES) C17H17N7O2S requires: 383. found: 384 (M+H)+.

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US09226929B2
Source dataset	uspto-grants-2016_01
ORD ID	ord-db2f1374c77744c380786e7863fc6c4b
Source note	uspto-grants-2016_01