2,4-Difluorophenylboronic acid → HCID 178527488, compound

Participants

Reaction Steps

The product was prepared according to General Procedure 3, described in Example 22, using 5-bromo-N-[3-(1H-tetrazol-5-yl)phenyl]thiophene-2-sulfonamide (Intermediate 17) (19 mg, 0.055 mmol) and 2,4-difluorophenylboronic acid (9 mg, 0.06 mmol). The title compound was obtained in 33% yield (6.9 mg). MS (ESI+) calcd mass for C17H11F2N5O2S2 419.032222, found 419.032372.

Provenance & Evidence