HuagongsheHuagongshe Chemistry Print Report · For research reference only
Methyl 4-(((1,1-dimethylethoxy)carbonyl)amino)-4-piperidinecarboxylate → {2-[4-(tert-Butoxycarbonylamino)-4-(methoxycarbonyl)piperidin-1-yl]pyrimidin-5-yl}-boronic acid
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Methyl 4-(((1,1-dimethylethoxy)carbonyl)amino)-4-piperidinecarboxylate | HCID 14537079 | — |
| Reactant | (2-Chloropyrimidin-5-yl)boronic acid | HCID 21747362 | — |
| Product | {2-[4-(tert-Butoxycarbonylamino)-4-(methoxycarbonyl)piperidin-1-yl]pyrimidin-5-yl}-boronic acid | HCID 131735241 | — |
Reaction Steps
The title compound was synthesised from methyl 4-(tert-butoxycarbonylamino)-piperidine-4-carboxylate and (2-chloropyrimidin-5-yl)boronic acid in accordance with General Method C.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09309243B2 |
| Source dataset | uspto-grants-2016_04 |
| ORD ID | ord-e87f36ca219b498786c36b99469d70c2 |
| Source note | uspto-grants-2016_04 |