Piperazin-2-one → HCID 118666134, compound

Participants

Reaction Steps

Synthesized from 3-(methylsulfinyl)-1-(5-phenylpyrimidin-2-yl)-1H-indole-6-carboxylic acid (200 mg, 0.53 mmol) and piperazin-2-one (64 mg, 0.63 mmol) in an analogous manner as described for example 52. White solid. Yield: 148 mg (61% of theory). HPLC-MS (method 4): Rt=2.6 min; m/z [M+H]+=460.3

Provenance & Evidence