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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 633832Generated: October 25, 2026

3-oxo-3,4-dihydro-2H-1,4-benzothiazine-6-carboxylic acid → HCID 71118894, compound

https://huagongshe.com/reaction/633832

Reaction equation

Participants

RoleNameHCIDCharge
Reactant3-oxo-3,4-dihydro-2H-1,4-benzothiazine-6-carboxylic acidHCID 760993—
Reactant1-Tert-butyl 2-methyl 4-aminopyrrolidine-1,2-dicarboxylateHCID 4913064—
Reactant3-bromomethyl-6-methoxy-3,4-dihydro-2H-1-thia-9-aza-phenanthreneHCID 86730711—
ProductHCID 71118894HCID 71118894—

Reaction Steps

The titled compound is prepared as an orange viscous oil following Scheme 1 and in analogy to Example 1 using 3-bromomethyl-6-methoxy-3,4-dihydro-2H-1-thia-9-aza-phenanthrene, 4-amino-pyrrolidine-1,2-dicarboxylic acid 1-tert-butyl ester 2-methyl ester and 3-oxo-3,4-dihydro-2H-benzo[1,4]thiazine-6-carboxylic acid as starting material.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09321788B2
Source datasetuspto-grants-2016_04
ORD IDord-52b482dc85ec4f39935a7dd782bed7e7
Source noteuspto-grants-2016_04