HRID641787

反应详情

EQUATION

反应方程式

HRID 641787 的结构方程式

PROCEDURE

实验过程

2.4 A solution of 50 mg of “A2” in 1 ml of formic acid (98-100%) is refluxed for 8 hours and subsequently purified via an RP18 column, giving 3 mg of 1-[4-(4-hydroxy-3H-imidazo[4,5-c]pyridin-2-ylmethyl)phenyl]-3-(2-fluoro-5-trifluoromethylphenyl)urea (“A3”), Rf 2.88.

WORKUP

后处理

  1. customsubsequently purified via an RP18 column