Hydrochloric Acid → HCID 86604121, compound

Participants

Reaction Steps

tert-Butyl 4-(3-{[(4-methylphenyl)sulfonyl]oxy}-1,2-benzisoxazol-5-yl)piperidine-1-carboxylate (285 mg, 0.603 mmol) was dissolved in anhydrous 4N HCl in dioxane (6 mL) and the resulting mixture was stirred at rt for 1 h. The reaction mixture was concentrated to afford 5-piperidin-4-yl-1,2-benzisoxazol-3-yl 4-methylbenzenesulfonate hydrochloride which did not require further purification.

Provenance & Evidence