HRID646440

反应详情

EQUATION

反应方程式

REACTANTS

反应物

HCID25236221

未命名化合物

结构：C[C@@H]1CCCN1C[C@@H]1CCCN1C(=O)c1ccc(B2OC(C)(C)C(C)(C)O2)cc1

HCID57980025

未命名化合物

PRODUCTS

生成物

结构：C[C@@H]1CCCN1C[C@@H]1CCCN1C(=O)c1ccc(-c2ccc(C(=O)N3CCCCC3)s2)cc1

HCID11605120

未命名化合物

收率 48%

PROCEDURE

实验过程

The title compound is prepared in a manner substantially analogous to General Procedure A using [2-(S)-(2-(R)-methyl-pyrrolidin-1-ylmethyl)-pyrrolidin-1-yl]-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-methanone (550 mg, 1.4 mmol) and (5-Bromo-thiophen-2-yl)-piperidin-1-yl-methanone (CAS 626242-11-3) (315 mg, 1.2 mmol) to give 260 mg (48% yield). MS (ES+) 466.2 (M+H)+

WORKUP

后处理

customto give 260 mg (48% yield)