Pyrazinecarbonyl chloride → N-Cyclopropyl-4-oxazol-5-yl-N-[1-(5-pyrazin-2-yl-[1,2,4]oxadiazol-3-yl)-piperidin-4-yl]-benzamide

Participants

Reaction Steps

The title compound is prepared from N-cyclopropyl-N-[1-(N-hydroxycarbamimidoyl)-piperidin-4-yl]-4-oxazol-5-yl-benzamide and pyrazine-2-carbonyl chloride following a procedure analogous to that described in Example 47. LC (method 2): tR=1.15 min; Mass spectrum (ESI+): m/z=458 [M+H]+.

Provenance & Evidence