6-[(S)-1-(tetrahydrofuran-2-yl)methoxy]isochromen-1-one → 4-(2-Methoxy-4-{1-oxo-6-[(S)-1-(tetrahydro-furan-2-yl)methoxy]-1H-isoquinolin-2-yl}-phenyl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	6-[(S)-1-(tetrahydrofuran-2-yl)methoxy]isochromen-1-one	HCID 66879690	—
Edukt	4-(4-Amino-2-methoxyphenyl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester	HCID 68987937	—
Produkt	4-(2-Methoxy-4-{1-oxo-6-[(S)-1-(tetrahydro-furan-2-yl)methoxy]-1H-isoquinolin-2-yl}-phenyl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester	HCID 68991497	—

Reaktionsschritte

Reaction of 6-[(S)-1-(Tetrahydro-furan-2-yl)methoxy]-isochromen-1-one with 4-(4-Amino-2-methoxy-phenyl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester by method AJ resulted in the desired product with the molecular weight of 549.67 (C31H39N3O6); MS (ESI): 550 (M+H+).

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US08822495B2
Quelldatensatz	uspto-grants-2014_09
ORD ID	ord-486c705217e54ff98f15dac07144bc8b
Quellennotiz	uspto-grants-2014_09