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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 712832Generated: October 30, 2026

1-benzylazetidine-2-carboxylic acid → HCID 71186307, compound

https://huagongshe.com/reaction/712832

Reaction equation

Participants

RoleNameHCIDCharge
Reactant1-benzylazetidine-2-carboxylic acidHCID 288936—
Reactant(S)-Methyl 4-(1-aminoethyl)benzoate hydrochlorideHCID 57462942—
ProductHCID 71186307HCID 7118630753.2%

Reaction Steps

The title compound (D76) (98 mg) was prepared according to the general procedure for amides preparation (Method C) starting from 1-benzylazetidine-2-carboxylic acid (100 mg, available from Apollo#OR7040) and (S)-methyl 4-(1-aminoethyl)benzoate hydrochloride (113 mg). Reaction time: 1 h

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS09181279B2
Source datasetuspto-grants-2015_11
ORD IDord-83f076cccdb742349530cc10143933be
Source noteuspto-grants-2015_11