反应详情

In analogy to the procedure described for the preparation of 4-(3-fluoro-4-trifluoromethyl-phenyl)-5,6-dihydro-[2]pyrindin-7-one (intermediate A-14 [C1]), replacing 4-(3-fluoro-4-trifluoromethyl-phenyl)-6,7-dihydro-5H-[2]pyrindine with 4-(4-trifluoromethyl-phenyl)-6,7-dihydro-5H-[2]pyrindine. The title compound was obtained as a light brown oil in 24% yield. MS: 278.1 (M+H+).