HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-Oxo-azetidine-1-carboxylic acid tert-butyl ester → HCID 67958091, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-Oxo-azetidine-1-carboxylic acid tert-butyl ester | HCID 1519404 | — |
| Reactant | 4-Amino-3-methylbenzotrifluoride | HCID 13750437 | — |
| Product | HCID 67958091 | HCID 67958091 | 21.4% |
Reaction Steps
The title compound (D32) (330 mg) was prepared according to the experimental procedure described in Description 30 starting from 1-Boc-3-azetidinone (800 mg, 4.67 mmol) and 4-Amino-3-methylbenzotrifluoride (818.4 mg, 4.67 mmol).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08828987B2 |
| Source dataset | uspto-grants-2014_09 |
| ORD ID | ord-dbd1b969ca3146dabb36fd51d7ef2a38 |
| Source note | uspto-grants-2014_09 |