4-Aminotetrahydropyran → HCID 24738511, compound

Participants

Reaction Steps

As described for Example 11b, 2-(5-methyl-3-phenyl-isoxazol-4-yl)-imidazo[1,2-a]pyridine-7-carboxylic acid (85 mg, 0.27 mmol) was converted, using 4-aminotetrahydropyran instead of aminomethylcyclopropane, to the title compound (61 mg, 57%) which was obtained as a yellow solid. MS: m/e=403.5 [M+H]+.

Provenance & Evidence