2-Methoxyethylamine → HCID 77750128, compound

HRID 840709Notes

Reaction equation

[CH2:1]([NH:3][C:4]([CH:6]1[CH2:10][CH:9]([N:11]2[C:15]3[N:16]=[C:17]([S:30][CH2:31][CH2:32][CH3:33])[N:18]=[C:19]([NH:20][CH:21]4[CH2:23][CH:22]4[C:24]4[CH:29]=[CH:28][CH:27]=[CH:26][CH:25]=4)[C:14]=3[N:13]=[N:12]2)[CH:8]([OH:34])[CH:7]1[OH:35])=[O:5])[CH3:2].[CH3:36][O:37]CCN>>[OH:35][CH:7]1[CH:8]([OH:34])[CH:9]([N:11]2[C:15]3[N:16]=[C:17]([S:30][CH2:31][CH2:32][CH3:33])[N:18]=[C:19]([NH:20][CH:21]4[CH2:23][CH:22]4[C:24]4[CH:25]=[CH:26][CH:27]=[CH:28][CH:29]=4)[C:14]=3[N:13]=[N:12]2)[CH2:10][CH:6]1[C:4]([NH:3][CH2:1][CH2:2][O:37][CH3:36])=[O:5]

Participants

Reactant 2

HCID 80182-Methoxyethylamine

HCID 77750217HCID 77750217, compound

Product 1

HCID 77750128HCID 77750128, compound

Procedure

The title compound was prepared according to the method of example 1, step d), using the product of example 1, step c) and 2-methoxyethylamine, followed by deprotection according to the method of example 1, step e).

Sources & evidence

ORD record: ord-cb616fe7c28a4424b632038479b36088
Source dataset: uspto-grants-2002_04
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US06369064B1

Reaction notes

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