2-Bromoanisole → HCID 59361538, compound
Reaction equation
[CH:1]1([N:9]2[C:12](=[O:13])[C:11]([CH3:15])([CH3:14])[NH:10]2)[CH2:8][CH2:7][CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1.Br[C:17]1[CH:22]=[CH:21][CH:20]=[CH:19][C:18]=1[O:23][CH3:24]>>[CH:1]1([N:9]2[C:12](=[O:13])[C:11]([CH3:15])([CH3:14])[N:10]2[C:17]2[CH:22]=[CH:21][CH:20]=[CH:19][C:18]=2[O:23][CH3:24])[CH2:8][CH2:7][CH2:6][CH2:5][CH2:4][CH2:3][CH2:2]1Participants
3
Procedure
2-Cyclooctyl-4,4-dimethyl-1,2-diazetidin-3-one prepared in Process 5 of Example 73 and 1-bromo-2-methoxybenzene was used for a similar reaction and treatment as Example 181, and the title compound was obtained as a pale yellow oil.
Workup
- customwas used for a similar reaction and treatment as Example 181
Sources & evidence
- ORD record
- ord-4d081bc9ebc541069a5940ac1d2448a0
- Source dataset
- uspto-grants-2012_08
- Patent number
- US08252781B2
Reaction notes
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