N-((4-(Aminosulphonyl)phenyl)methyl)acetamide → N-[4-({[({2-[4-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)phenyl]ethyl}amino)carbonyl]amino}sulfonyl)benzyl]acetamide

Participants

Reaction Steps

The title compound was prepared according to the procedure described in step 1 of Example 42 from phenyl 2-[4-(3,5-dimethyl-4-phenyl-1H-pyrazol-1-yl)phenyl]ethylcarbamate (step 1 of Example 22) and N-[4-(aminosulfonyl)benzyl]acetamide: 1H-NMR [CDCl3/CD3OD(4:1)]δ 7.90-7.87 (2H, m), 7.48-7.26 (11H, m), 4.44 (2H, s), 3.45-3.41 (2H, m), 2.87-2.82 (2H, m), 2.32 (3H, s), 2.27 (3H, s), 2.03 (3H, s).

Provenance & Evidence