HuagongsheHuagongshe Chemistry Print Report · For research reference only
4-(2-Carboxyethyl)benzeneboronic acid → 3-{4-[6-Amino-5-(pyridin-4-ylcarbamoyl)-pyridin-3-yl]-phenyl}-propionic acid
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 4-(2-Carboxyethyl)benzeneboronic acid | HCID 3863484 | — |
| Reactant | 2-amino-5-bromo-N-(pyridin-4-yl)nicotinamide | HCID 62155416 | — |
| Product | 3-{4-[6-Amino-5-(pyridin-4-ylcarbamoyl)-pyridin-3-yl]-phenyl}-propionic acid | HCID 71061007 | — |
Reaction Steps
Reaction of 2-amino-5-bromo-N-pyridin-4-yl-nicotinamide with 3-(4-boronophenyl)-propanoic acid gives the compound “A32”; HPLC/MS: 1.28 min, [M+H]=363;
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09273029B2 |
| Source dataset | uspto-grants-2016_03 |
| ORD ID | ord-baafaa84b97646d19902aac9e181ba32 |
| Source note | uspto-grants-2016_03 |