反应详情

The title compound is prepared according to the procedure of Example 2, Step 3, except that 4-(3-chloropropoxy)-1H-indole is used in place of 4-(2-chloro-ethoxy)-1H-indole and 3-(3,4-dichloro-phenyl)-8-aza-bicyclo[3.2.1]oct-2-ene is used in place of 3-(8-aza-bicyclo[3.2.1]oct-2-en-3-yl)-1H-indole. The corresponding oxalate salt is prepared by treating the title compound with 1 equiv. of oxalic acid in EtOH. Yield: 22% of an off-white solid. mp: 150-153° C.; MS (ES) m/z: 427.2 (MH)+.

1. customThe title compound is prepared
2. customThe corresponding oxalate salt is prepared