[F:1][C:2]1[CH:3]=[CH:4][C:5]2[S:9][C:8](C)=[N:7][C:6]=2[CH:11]=1.[OH-].[Na+]>C(O)CO>[F:1][C:2]1[CH:3]=[CH:4][C:5]([S:9][CH3:8])=[C:6]([CH:11]=1)[NH2:7]5-Fluoro-2-methylbenzothiazole was heated with ethylene glycol and 10N sodium hydroxide solution and the resulting thiol methylated using procedures similar to those described in Example 5, to give 5-fluoro-2-(methylthio)aniline.
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