Benzenamine, 4-(4-morpholinyl)- → HCID 87319734, compound

HRID 1470975Notes

Reaction equation

HRID 1470975 reaction equation
CS(O[C@H:6]([C:24]1[CH:29]=[CH:28][C:27]([N+:30]([O-:32])=[O:31])=[CH:26][CH:25]=1)[CH2:7][CH2:8][C@H:9](OS(C)(=O)=O)[C:10]1[CH:15]=[CH:14][C:13]([N+:16]([O-:18])=[O:17])=[CH:12][CH:11]=1)(=O)=O.[O:33]1[CH2:38][CH2:37][N:36]([C:39]2[CH:45]=[CH:44][C:42]([NH2:43])=[CH:41][CH:40]=2)[CH2:35][CH2:34]1>CN1C(=O)CCC1>[N+:16]([C:13]1[CH:14]=[CH:15][C:10]([C@H:9]2[CH2:8][CH2:7][C@H:6]([C:24]3[CH:29]=[CH:28][C:27]([N+:30]([O-:32])=[O:31])=[CH:26][CH:25]=3)[N:43]2[C:42]2[CH:41]=[CH:40][C:39]([N:36]3[CH2:37][CH2:38][O:33][CH2:34][CH2:35]3)=[CH:45][CH:44]=2)=[CH:11][CH:12]=1)([O-:18])=[O:17]

Participants

4

Reactant 2

HCID 75655Benzenamine, 4-(4-morpholinyl)-HCID 87378855HCID 87378855, compound

Product 1

HCID 87319734HCID 87319734, compound

Reagents, catalysts & solvents 1

HCID 13387N-methyl-2-pyrrolidoneSolvent

Procedure

The product from Example 38A and 4-morpholinoaniline were processed using the method described in Example 1D using NMP for the solvent to afford the title compound. MS (ESI) m/z 475 (M+H)+.

Sources & evidence

ORD record
ord-f7a272302d86426b8f3026782f1d2329
Source dataset
uspto-grants-2015_04
Patent number
US09006387B2

Reaction notes

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