2-Methylpyridine → 2-Methylpyridine-4-boronic acid pinacol ester

HRID 1490475Notes

Reaction equation

HRID 1490475 reaction equation
Cc1ccccn1>CC1(C)OB(B2OC(C)(C)C(C)(C)O2)OC1(C)C.C1CCOC1>Cc1cc(B2OC(C)(C)C(C)(C)O2)ccn1

Participants

4

Reactant 1

HCID 79752-Methylpyridine

Product 1

HCID 164142742-Methylpyridine-4-boronic acid pinacol esterYield 92%

Reagents, catalysts & solvents 2

HCID 2733548Bis(pinacolato)diboraneReagentHCID 8028TetrahydrofuranSolvent

Conditions

Temperature
80 °C

Sources & evidence

ORD record
ord-743548bea2e0400c88996cd6a1e0177c
Source dataset
Borylation dataset from Roche

Reaction notes

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