HRID1490506

反应详情

EQUATION

反应方程式

HRID 1490506 的结构方程式

AUXILIARIES

试剂、催化剂与溶剂

5

CONDITIONS

反应条件

温度
120 °C

PROCEDURE

实验过程

Prepared from 5-fluoro-N-(triisopropylsilyl)-1H-indole (4f, 58.3 mg, 0.200 mmol, 1.00 equiv) and catBH (96.0 mg, 0.800 mmol, 4.00 equiv) according to GP 2. The title compound was purified by flash column chromatography using cyclohexane/EtOAc/Et3N (30/1/1) as eluent to afford 6f (44.5 mg, 53%) as a white foam.