HCID 19803507, compound → HCID 19803565, compound

HRID 1682075Notes

Reaction equation

HRID 1682075 reaction equation
[NH:1]1[CH2:6][CH2:5][CH2:4][CH:3]([CH2:7][N:8]2[CH2:16][C:15]3[C:10](=[CH:11][C:12]([O:19][CH3:20])=[C:13]([O:17][CH3:18])[CH:14]=3)[C:9]2=[O:21])[CH2:2]1.C1(S(O[CH2:32][CH2:33][CH2:34][C:35]2[C:43]3[C:38](=[CH:39][CH:40]=[CH:41][CH:42]=3)[NH:37][CH:36]=2)(=O)=O)C=CC=CC=1>CN(C)C=O.C(N(CC)CC)C>[NH:37]1[C:38]2[C:43](=[CH:42][CH:41]=[CH:40][CH:39]=2)[C:35]([CH2:34][CH2:33][CH2:32][N:1]2[CH2:6][CH2:5][CH2:4][CH:3]([CH2:7][N:8]3[CH2:16][C:15]4[C:10](=[CH:11][C:12]([O:19][CH3:20])=[C:13]([O:17][CH3:18])[CH:14]=4)[C:9]3=[O:21])[CH2:2]2)=[CH:36]1

Participants

5

Reactant 2

HCID 19803507HCID 19803507, compoundHCID 19803590HCID 19803590, compound

Product 1

HCID 19803565HCID 19803565, compound

Reagents, catalysts & solvents 2

HCID 6228DimethylformamideSolventHCID 8471TriethylamineSolvent

Procedure

Prepared from 2-[(piperidin-3-yl)-methyl]-5,6-dimethoxy-1-oxo-1,3-dihydro-isoindole and 3-(3-benzenesulphonyloxy-propyl)-indole in dimethylformamide and triethylamine analogously to Example 1.

Sources & evidence

ORD record
ord-468d71274ccb4872b97642f363620fe4
Source dataset
uspto-grants-1992_12
Patent number
US05175157

Reaction notes

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