反应详情

In analogy to the procedure described in example 1.2, cyclohexyl-(2-phenyl-2H-indazol-3-yl)-amine (example 1.1) was reacted with (3-fluoro-4-isocyanato-phenoxy)-acetic acid methyl ester in 1,2-dichloroethane in the presence of Et3N (1.4 eq.) for 2 days under reflux conditions to give the title compound as yellow solid. MS: m/e=516.8 [M+H+].