HRID1796636

反应详情

EQUATION

反应方程式

HRID 1796636 的结构方程式

AUXILIARIES

试剂、催化剂与溶剂

2

PROCEDURE

实验过程

To a solution of 397A (32 mg, 0.090 mmol) in CH2Cl2 (1 ml) was added Tf2O (18 μl, 0.099 mmol) at −10° C. The reaction mixture was stirred for 5 min, diluted with EtOAc, washed with brine, dried and concentrated to give 397 (42 mg, 95%) LCMS Found: (M+H)+=489.0

WORKUP

后处理

  1. washwashed with brine
  2. customdried
  3. concentrationconcentrated