反应详情

In the similar fashion using route 14 general procedure 27, 7-methyl-8-aminoquinoline (200 mg, 1.26 mmol), benzenesulfonyl chloride (260 mg, 1.5 mmol) and DMAP (cat.) gave the title compound (250 mg, 67%) after purification by column chromatography with DCM as the eluent.