反应详情

The title compound was prepared in analogy to the compound of Example 236 using a 2 M solution of methylamine in MeOH instead of pyrrolidine (tR 2.61 min (conditions 3), MH+=384.3, 1H-NMR in DMSO-d6: 8.82 (m, 1H); 8.56 (s, 1H); 8.32 (m, 1H); 8.19 (s, 2H); 8.11 (d, 1H); 7.94 (m, 2H); 7.78 (m, 1H); 7.66 (s, 1H); 7.54 (d, 1H); 7.48 (dd, 1H); 4.53 (m, 4H); 3.40 (t, 2H); 2.55 (s, 3H)).