Anthranilic Acid → HCID 11626464, compound
Reaction equation
[C:1]([OH:10])(=O)[C:2]1[C:3](=[CH:5][CH:6]=[CH:7][CH:8]=1)[NH2:4].[F:11][C:12]([F:16])([F:15])[CH2:13][NH2:14].[CH:17](=O)[C:18]1[CH:23]=[CH:22][C:21]([O:24][CH3:25])=[CH:20][CH:19]=1.Cl[CH2:28][CH2:29][CH2:30]Br.[NH:32]1[CH2:37][CH2:36]C[CH2:34][CH2:33]1>>[N:32]1([CH2:37][CH2:36][CH2:25][O:24][C:21]2[CH:22]=[CH:23][C:18]([C:17]3[N:14]([CH2:13][C:12]([F:16])([F:15])[F:11])[C:1](=[O:10])[C:2]4[C:3](=[CH:5][CH:6]=[CH:7][CH:8]=4)[N:4]=3)=[CH:19][CH:20]=2)[CH2:33][CH2:34][CH2:30][CH2:29][CH2:28]1Participants
6
Procedure
The entitled compound was obtained according to the method of Example 1 but starting from anthranilic acid, 2,2,2-trifluoroethylamine, 4-anisaldehyde, 1-chloro-3-bromopropane and piperidine.
Workup
- customThe entitled compound was obtained
Sources & evidence
- ORD record
- ord-d0c45b6bcf834e2e9966c591db05d28f
- Source dataset
- uspto-grants-2011_06
- Patent number
- US07960394B2
Reaction notes
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