反应详情

To a suspension of compound AE or AM′ (1.0 equiv.) in DMF, DIC (1.5 equiv.) or EDCI (1.5 equiv.), HOBt (1.5 equiv.) and the selected amine (1.5-5.0 equiv.) were added. The mixture was stirred at R.T. for 12-72 Hrs or heated through microwave irradiation for 5 min at 150° C.

1. temperatureheated through microwave irradiation for 5 min at 150° C.